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Rifampin
Rifampin :
Antibiotic ID :
UD0038
Full Name :
Rifampin
Synonyms :
Rifampicin, Rifadin, Rimactane, Rimactan, Rifamycin AMP, Rifampicinum, Riforal, Tubocin, Rifa
Class :
Beta Lactum
Chemical Description :
Molecular Formula :
C
43
H
58
N
4
O
12
Molecular Weight :
822.94022
InChIKey :
FZYOVNIOYYPUPY-ZTWDQPHTSA-N
IUPAC Name :
NA
Structural Description :
Canonical SMILES :
CC1C=CC=C(C(=O)NC2=C(C3=C(C(=C4C(=C3C(=O)C2=CNN5CCN(CC5)C)C(=O)C(O4)(OC=CC(C(C(C(C(C(C1O)C)O)C)OC(=O)C)C)OC)C)C)O)O)C
Isomeric SMILES :
C[C@H]1/C=C/C=C(\C(=O)NC\2=C(C3=C(C(=C4C(=C3C(=O)/C2=C/NN5CCN(CC5)C)C(=O)[C@](O4)(O/C=C/[C@@H]([C@H]([C@H]([C@@H]([C@@H]([C@@H]([C@H]1O)C)O)C)OC(=O)C)C)OC)C)C)O)O)/C
2D Structure :
2D
3D Structure :
3D
SDF :
SDF file
Fuctional Description :
Rifampin Target :
A semisynthetic antibiotic produced from Streptomyces mediterranei. It has a broad antibacterial spectrum, including activity against several forms of Mycobacterium. In susceptible organisms it inhibits DNA-dependent RNA polymerase activity by forming a stable complex with the enzyme. It thus suppresses the initiation of RNA synthesis. Rifampin is bactericidal, and acts on both intracellular and extracellular organisms
(MeSH)
.
KEGG :
D00211
DRUG BANK :
DB01045
Pub Chem CID :
5381226
Antibiotics Resistance Reports :
Upregulators :
Gene :
mfdA
Downregulators :
NA
Note :
NA* - Not Available
Bibliography :
MdfA, an Escherichia coli multidrug resistance protein with an extraordinarily broad spectrum of drug recognition
, Edgar R, Bibi E.
, Journal of Bactriology
, 1997,
179
(7): 2274-80.
PMID:
9079913.